Cabergoline is a medication used to treat high prolactin levels caused by the use of steroids such as trenbolone and nandrolone. It is particularly useful for women as it can restore fertility.
This medicine can cause dizziness. Be careful driving or using machinery until you know how it affects you.
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What is Cabergoline?
Cabergoline, also know as Dostinex, is a medication used to treat hyperprolactinemia (high levels of prolactin in the body). It works by blocking dopamine receptors in the brain, preventing the release of the prolactin hormone. It can be taken by mouth or by injection. The dosage of Cabergoline will depend on your condition and other factors. For example, in men, it can be used to reduce symptoms of high prolactin levels such as breast enlargement, nipple discharge, low body hair, reduced muscle mass, and decreased libido. In addition, it can help to increase the quality and volume of seminal fluid.
In clinical trials, this drug has bee shown to be effective in treating both idiopathic hyperprolactinemia and micro- or macroprolactinomas. It has a low toxicity, is well tolerant, and has few side effects. It can be use as a stand-alone treatment or in combination with other medications such as levothyroxine, methotrexate, or glucocorticoids.
Although this drug is safe for most people, it is not recommend for pregnant women or breastfeeding mothers. It may also cause a condition called fibrosis, which is when the tissue in your body scars and hardens. This can happen in the lungs or around your heart, and it can be dangerous. It is important to tell your doctor if you have any history of fibrosis before starting this medication.
Another potential side effect of this medication is depression. This can occur in up to 20% of patients taking this drug. If you experience depression while taking Cabergoline Bodybuilding, you should talk to your doctor about it.
This medication may also increase your risk of developing gambling problems or other intense urges or behaviors that are unusual for you. It is important to tell your doctor unless you are comfortable discussing these issues with him or her.
This medication should not be take if you are allergic to it or any other ergot medicine, have a history of heart valve disease, or have uncontrolled high blood pressure or liver disease. It is also not recommend for use by elderly adults or those with a history of seizures.
How Does Cabergoline Work?
Cabergoline works by blocking the release of prolactin from the pituitary gland. This reduces the amount of breast milk a woman produces and may also help with other problems caused by high levels of prolactin, such as changes in the menstrual cycle or sex drive. Cabergoline can also increase testosterone in males with hyperprolactinemia, which may improve erectile function and fertility.
Cabergoline is available in tablet form to take by mouth, usually two times a week. It is important to take it exactly as prescribed by your doctor. Read the directions on your prescription label carefully, and ask your doctor or pharmacist to explain any part you do not understand. Take the medicine with or without food as directed. Your doctor will probably start you on a low dose and gradually increase your dose, not more often than every four weeks.
When you first start taking this medicine, it may make you sleepy. It is important not to drive or use machines until you know how this drug affects you. Your doctor will check your heart and lung function from time to time while you are taking this medication.
Women taking this drug should not get pregnant while they are taking it and for one month after they stop. They should use nonhormonal birth control (such as barrier methods or condoms) and tell their doctors if they become pregnant during treatment. Women with microprolactinomas can sometimes get pregnant while they are taking cabergoline. However, women with macroprolactinomas are not likely to be able to conceive even while they are taking this drug.
What are the Side Effects of Cabergoline?
Cabergoline is a drug that has bee found to reduce prolactin secretion in the pituitary gland of animals and humans. It works by binding to the dopamine receptors and blocking their activation. Moreover, it does not have significant affinity for dopamine D1 and adrenergic receptors or 5-HT1- and 5-HT2 serotonin receptors, so it doesn’t affect the levels of these hormones in the body.
During the first few weeks of treatment, some people may experience mild side effects, such as dizziness or stomach upset. These should pass as the body gets used to the medicine. If the symptoms get worse or persist, talk to your doctor. They may be able to offer advice on how to help reduce these side effects.
It is recommend that you take the tablets with food, as this may decrease the likelihood of stomach upset. You should also avoid taking other drugs which may interact with this medication. For example, erythromycin or clarithromycin (types of antibiotics) can increase the levels of cabergoline in the body, and it is important not to take these with this drug. Similarly, other drugs such as domperidone and metoclopramide can counteract the effect of this medication, so you should avoid these.
If you have been taking cabergoline for a long time, your endocrinologist will monitor you regularly, with blood tests and repeated pituitary MRI scans. This will enable them to see whether the treatment is working, and if it is safe to stop it.
Your doctor will tell you how often to take the drug and how much, depending on your condition. You may need to take it just for a few days, if you are trying to suppress breast milk; or each day, if you have Parkinson’s disease; or it may be a long-term treatment to lower your prolactin levels.
What is the Dosage of Cabergoline?
Dosage is tailore to each patient based on their prolactin levels and the symptoms they are experiencing. It is usually start with a low dose (0.025 mg per day) take by mouth on two days of the week to reduce stomach upset, and gradually increased over 4 weeks to the target dose of between 0.5 and 1 mg twice weekly. Your endocrinologist will monitor your blood prolactin level and pituitary MRI scans during this time. They will use these to check for shrinkage of the prolactin-producing tumours and to determine whether you need to be switcher to a different medication.
Unlike the older drugs use to treat hyperprolactinemia, such as bromocriptine, cabergoline has a long duration of action and does not nee to be taken as frequently. It is also more effective than other ergot derivatives in lowering PRL and in causing tumor shrinkage. In addition, it is not associate with the same spectrum of psychiatric side effects as other dopamine agonists.
This medication is not recommende in pregnancy, as it can harm a unborn baby. It is also not recommende for women who are breastfeeding, as it can pass into breast milk and affect the baby. Cabergoline is also not recommende for anyone who has a history of heart and lung diseases, liver disease, or certain other types of tumors Read More.
